COMPETITIVE INHIBITION OF PROCAINE CONVULSIONS BY ITS SPLIT-PRODUCTS
نویسندگان
چکیده
منابع مشابه
Competitive inhibition of calcineurin phosphatase activity by its autoinhibitory domain.
Calcineurin (protein phosphatase 2B), a calmodulin- and calcium-dependent serine/threonine phosphatase, appears to be regulated by a C-terminal autoinhibitory domain. A 25 amino acid peptide derived from this domain inhibits calcineurin phosphatase activity in vitro. Here we show that a 97 amino acid fragment of the calcineurin A alpha C-terminus is approx. 8-fold more potent than the shorter p...
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ژورنال
عنوان ژورنال: Journal of Biological Chemistry
سال: 1945
ISSN: 0021-9258
DOI: 10.1016/s0021-9258(19)51323-0